SCHEMBL7320134

SCHEMBL7320134

O=C(N[C@@H](Cc1ccccc1)C(=O)O)OCc1ccccc1.O=CCCl

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.58
ITGA2B P08514 6/20 0.58
TACR1 P25103 2/20 0.58
CTSL P07711 4/20 0.57
CTSB P07858 4/20 0.57
CTSS P25774 2/20 0.57
CTSK P43235 1/20 0.57
ALDH1A1 P00352 1/20 0.56
ALOX15 P16050 1/20 0.56
MME P08473 1/20 0.55
ECE1 P42892 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9127701 1.00 ITGB3 (0.58) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL7366118 0.91 TACR1 (0.62) ITGB3ITGA2BTACR1CTSLCTSB
Hypochlorous Acid SCHEMBL7368156 0.90 TACR1 (0.65) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL220648 0.90 TACR1 (0.68) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL479010 0.90 TACR1 (0.68) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL7372270 0.90 TACR1 (0.68) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL219151 0.90 TACR1 (0.68) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL26661077 0.90 TACR1 (0.68) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL7318252 0.90 ITGB3 (0.58) ITGB3ITGA2BTACR1CTSLCTSB
SCHEMBL9127693 0.88 ITGB3 (0.60) ITGB3ITGA2BTACR1CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999059989-A1 PROCESS FOR THE PREPARATION OF A BENZO FUSED HETEROCYCLO SULFONYL HALIDE INTERMEDIATE G.D. SEARLE & CO. (US) 1999-11-25 WO disclosed
EP-0769936-A1 SELF-EMULSIFYING DRUG DELIVERY SYSTEM G.D. SEARLE & CO. (US) 1997-05-02 EP disclosed
WO-1996003113-A1 SELF-EMULSIFYING DRUG DELIVERY SYSTEM G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed
EP-0677048-A1 CYCLIC SULFONE CONTAINING RETROVIRAL PROTEASE INHIBITORS. SEARLE & CO (US) 1995-10-18 EP disclosed
EP-0641325-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1995-03-08 EP disclosed
WO-1995006061-A1 RETROVIRAL PROTEASE INHIBITORS AND COMBINATIONS THEREOF G.D. SEARLE & CO. (US) 1995-03-02 WO disclosed
WO-1994014793-A1 CYCLIC SULFONE CONTAINING RETROVIRAL PROTEASE INHIBITORS G. D. SEARLE & CO. (US) 1994-07-07 WO disclosed
EP-0558630-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1993-09-08 EP disclosed
EP-0554400-A1 RETROVIRAL PROTEASE INHIBITORS. MONSANTO CO (US) 1993-08-11 EP disclosed
WO-1992008701-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed
WO-1992008698-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed
US-4670541-A Use of diamino alcohols as analgesic agents E. R. SQUIBB & SONS, INC. (US) 1987-06-02 US disclosed
US-4552866-A Use of diamino alcohols as analgesic agents E. R. SQUIBB & SONS, INC. (US) 1985-11-12 US disclosed