SCHEMBL7320136

SCHEMBL7320136

CCCCCCN(CCC(C)COS(=O)(=O)c1ccc(C)cc1)S(=O)(=O)c1cccc2cnccc12

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.44
ROCK1 Q13464 8/20 0.44
P2RX7 Q99572 8/20 0.42
NR3C1 P04150 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
CAMK2D Q13557 1/20 0.37
P2RX4 Q99571 1/20 0.37
CAMK2A Q9UQM7 1/20 0.37
F2 P00734 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10496397 0.90 P2RX7 (0.43) ROCK2ROCK1P2RX7NR3C1ALDH1A1
SCHEMBL7327226 0.88 ROCK2 (0.48) ROCK2ROCK1P2RX7LMNAF2
SCHEMBL7319421 0.88 ROCK2 (0.48) ROCK2ROCK1P2RX7LMNAF2
SCHEMBL10496402 0.88 ROCK2 (0.48) ROCK2ROCK1P2RX7LMNAF2
SCHEMBL7316438 0.88 ROCK2 (0.48) ROCK2ROCK1P2RX7LMNAF2
SCHEMBL7322591 0.86 ROCK2 (0.45) ROCK2ROCK1P2RX7NR3C1LMNA
SCHEMBL7326031 0.86 ROCK2 (0.46) ROCK2ROCK1P2RX7NR3C1LMNA
SCHEMBL10496387 0.85 ROCK2 (0.42) ROCK2ROCK1P2RX7NR3C1LMNA
SCHEMBL7322056 0.85 P2RX7 (0.44) ROCK2ROCK1P2RX7NR3C1ALDH1A1
SCHEMBL10496437 0.84 ROCK2 (0.43) ROCK2ROCK1P2RX7LMNAF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0287696-B1 ISOQUINOLINE DERIVATIVES Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1991-01-02 EP disclosed
US-4798897-A (AMINOALKYL)AMINOSULFONYL-SUBSTITUTED CARDIOVASCULAR AND RESPIRATORY SYSTEM DISORDERS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1989-01-17 US disclosed
EP-0287696-A1 Isoquinoline derivatives Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1988-10-26 EP disclosed