SCHEMBL7320464

SCHEMBL7320464

COc1ccc(I)c(CCC(C)N(C)C(=O)Cc2ccc(OC)c(OC)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
LMNA P02545 4/20 0.46
HTT P42858 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPC1 O15118 1/20 0.45
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
MAPT P10636 3/20 0.40
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GLA P06280 1/20 0.40
STAT3 P40763 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LTB4R Q15722 2/20 0.39
LTB4R2 Q9NPC1 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7322670 0.81 CYP3A4 (0.48) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL9158055 0.77 OPRD1 (0.49) MEN1KMT2ALMNAHTTSMN1; SMN2
SCHEMBL9160427 0.76 OPRD1 (0.48) MEN1KMT2ALMNAHTTNPC1
SCHEMBL7325376 0.76 CDK8 (0.61) MEN1KMT2ALMNAHTTSMN1; SMN2
Oxalic Acid SCHEMBL10689687 0.75 MEN1 (0.50) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL10411173 0.75 AOC3 (0.40)
SCHEMBL10687447 0.73 CYP3A4 (0.49) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7313447 0.70 CYP3A4 (0.62) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7323259 0.69 SMN1; SMN2 (0.56) MEN1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL7315866 0.69 HTR2A (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0250254-B1 CIS & TRANS STILBENES AND THEIR COMPOSITION FOR THE TREATMENT OF HYPERTENSION McNeilab, Inc. (US) 1991-06-19 EP disclosed
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
EP-0250254-A1 Cis & trans stilbenes and their composition for the treatment of hypertension McNeilab, Inc. (US) 1987-12-23 EP disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed