SCHEMBL7323259

SCHEMBL7323259

COc1ccc(I)c(CCNCCc2ccc(OC)c(OC)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.56
POLB P06746 1/20 0.52
ATM Q13315 1/20 0.52
ALDH1A1 P00352 3/20 0.50
KDM4E B2RXH2 2/20 0.50
GLA P06280 1/20 0.50
KMT2A Q03164 3/20 0.49
MEN1 O00255 1/20 0.49
SLC2A1 P11166 1/20 0.49
MAPT P10636 3/20 0.48
SMPD1 P17405 1/20 0.48
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
ALOX15 P16050 1/20 0.46
ADRB2 P07550 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA5A P35218 1/20 0.46
CA9 Q16790 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22222297 0.83 KMT2A (0.66) SMN1; SMN2POLBATMALDH1A1KDM4E
SCHEMBL9825369 0.82 KCNH2 (0.50) SMN1; SMN2POLBATMKMT2AMEN1
SCHEMBL7435099 0.81 ATM (0.76) SMN1; SMN2POLBATMALDH1A1KDM4E
Hydrochloric Acid SCHEMBL7320769 0.81 KCNH2 (0.49) SMN1; SMN2POLBATMKMT2AMEN1
Hydrochloric Acid SCHEMBL11808765 0.80 ATM (0.73) SMN1; SMN2POLBATMALDH1A1KDM4E
SCHEMBL9689514 0.78 CA1 (0.65) SMN1; SMN2POLBATMALDH1A1KDM4E
SCHEMBL7313447 0.78 CYP3A4 (0.62) SMN1; SMN2ALDH1A1KDM4EKMT2AMEN1
SCHEMBL4103249 0.77 KDM4E (0.74) SMN1; SMN2POLBATMALDH1A1KDM4E
SCHEMBL7320574 0.77 SLC2A1 (0.50) SMN1; SMN2POLBATMALDH1A1KMT2A
Perchlorate SCHEMBL7325314 0.76 HTR2A (0.47) POLBATMALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed