SCHEMBL7320574

SCHEMBL7320574

COc1ccc(C#Cc2ccccc2)c(CCNCCc2ccc(OC)c(OC)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.50
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
ADRB2 P07550 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
SMPD1 P17405 1/20 0.47
ADRB1 P08588 2/20 0.45
ADRB3 P13945 2/20 0.45
ALDH1A1 P00352 1/20 0.45
ALOX15 P16050 1/20 0.45
KMT2A Q03164 2/20 0.44
BCHE P06276 1/20 0.44
POLB P06746 1/20 0.44
ATM Q13315 1/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210269 0.88 HTT (0.47) SLC2A1MTNR1AMTNR1BADRB2SMN1; SMN2
SCHEMBL9824451 0.85 SLC2A1 (0.52) SLC2A1MTNR1AMTNR1BADRB2SMN1; SMN2
SCHEMBL7321263 0.84 CYP1A2 (0.55) SMN1; SMN2SMPD1ALDH1A1KMT2AMEN1
SCHEMBL7314273 0.83 MTNR1B (0.55) SLC2A1MTNR1AMTNR1BSIGMAR1KMT2A
SCHEMBL10593444 0.80 KMT2A (0.62) ADRB2ADRB1ADRB3KMT2AATM
Hydrochloric Acid SCHEMBL7323113 0.80 SMPD1 (0.55) MTNR1AMTNR1BSMN1; SMN2SMPD1KMT2A
SCHEMBL9218599 0.79 CYP1A2 (0.41) MTNR1AMTNR1BSIGMAR1SMPD1ALDH1A1
Hydrochloric Acid SCHEMBL7311252 0.78 BLM (0.42) MTNR1AMTNR1BSIGMAR1SMPD1ALDH1A1
SCHEMBL7318305 0.78 SMPD1 (0.43) SIGMAR1SMPD1ALDH1A1KMT2AMEN1
Fumaric Acid SCHEMBL7356000 0.78 CYP3A4 (0.47) MTNR1AMTNR1BSMPD1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed