SCHEMBL7322803

SCHEMBL7322803

CCCCN1CCC(Cc2cccc3ccc(=O)n(C(=O)O)c23)CC1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.45
RAB9A P51151 1/20 0.42
HTR7 P34969 4/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346871 0.83 KCNH2 (0.46) KCNH2RAB9ADRD4
SCHEMBL7357788 0.80 HTR7 (0.55) KCNH2RAB9AHTR7
SCHEMBL27416355 0.74 KCNH2 (0.45) KCNH2RAB9ADRD4
SCHEMBL7383392 0.74 KCNH2 (0.51) KCNH2HTR7DRD4
SCHEMBL7346867 0.73 SLC6A2 (0.46) KCNH2RAB9ASLC6A2SLC6A4
SCHEMBL7324117 0.73 CHRM1 (0.48) KCNH2RAB9ADRD4
SCHEMBL7348366 0.72 KCNH2 (0.46) KCNH2RAB9ADRD4
Hydrochloric Acid SCHEMBL7533243 0.72 HTR7 (0.41) KCNH2RAB9AHTR7
Hydrochloric Acid SCHEMBL7537449 0.71 HTR7 (0.40) KCNH2RAB9AHTR7
SCHEMBL7346874 0.70 KCNH2 (0.46) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708174-A Heterocyclic-esters or -amides used as 5-HT4 receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 1998-01-13 US claimed
WO-1994008994-A1 HETEROCYCLIC -ESTERS OR -AMIDES USED AS 5-HT4 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-28 WO claimed
US-5708174-A Heterocyclic-esters or -amides used as 5-HT4 receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 1998-01-13 US disclosed