SCHEMBL7322912

SCHEMBL7322912

COC(=O)[C@H](CC(C)C)NC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 10/20 0.52
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
ACE P12821 1/20 0.47
CMA1 P23946 1/20 0.47
CAPN1 P07384 2/20 0.45
REN P00797 1/20 0.45
CTSK P43235 3/20 0.44
CTSL P07711 2/20 0.44
CTSS P25774 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7322906 1.00 FKBP1A (0.52) FKBP1AALDH1A1CYP3A4TSHRACE
SCHEMBL28051124 0.86 CMA1 (0.57) CMA1CAPN1RENCTSKCTSL
SCHEMBL1992452 0.85 FKBP1A (0.60) FKBP1AALDH1A1CYP3A4TSHRCMA1
SCHEMBL7320486 0.84 SMN1; SMN2 (0.48) ACEREN
SCHEMBL7320499 0.84 SMN1; SMN2 (0.48) ACEREN
SCHEMBL13413313 0.83 FKBP1A (0.51) FKBP1AACERENCTSKCTSL
SCHEMBL28349215 0.82 FKBP1A (0.56) FKBP1AACERENCTSKCTSL
SCHEMBL13413249 0.82 FKBP1A (0.58) FKBP1AACERENCTSKCTSL
SCHEMBL13413216 0.82 FKBP1A (0.53) FKBP1AACERENCTSKCTSL
SCHEMBL30051146 0.81 ALDH1A1 (0.62) FKBP1AALDH1A1CYP3A4TSHRACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4691007-A HUMAN LEUKOCYTE ELASTASE INHIBITORS ICI AMERICAS INC. (US) 1987-09-01 US disclosed
US-4596789-A Pharmaceuticals ICI AMERICAS INC. (US) 1986-06-24 US disclosed
EP-0124317-A2 Proline derivatives ICI AMERICAS INC. (US) 1984-11-07 EP disclosed