SCHEMBL7323015

SCHEMBL7323015

Cc1nc(C)c([N+](=O)[O-])[nH]1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.46
ALDH1A1 P00352 5/20 0.46
GAA P10253 2/20 0.42
MDM2 Q00987 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.39
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
GFER P55789 1/20 0.35
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11754489 0.80 MAPT (0.36) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL9762507 0.80 MAPT (0.39) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL29105506 0.80 MAPT (0.36) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL8953652 0.79 MAPT (0.45) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL10487044 0.77 MAPT (0.47) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL8342993 0.77 ALDH1A1 (0.44) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL11405760 0.77 MAPT (0.44) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL29105510 0.77 ALDH1A1 (0.41) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL11077687 0.77 ALDH1A1 (0.34) MAPTALDH1A1GAAMDM2SMN1; SMN2
SCHEMBL29105514 0.77 GFER (0.35) MAPTALDH1A1GAAMDM2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116813553-A Selective deuterated N-methylation method of polyazaaromatic compound 四川大学 2023-09-29 CN disclosed
CN-105829433-A CROSSLINKABLE NITRILE RUBBER COMPOSITION AND RUBBER CROSSLINKED PRODUCT 日本瑞翁株式会社 2016-08-03 CN disclosed
CN-1035824-A The preparation method of 1-alkyl-5-nitroimidazole RHONE POULENC SANTE (FR) 1989-09-27 CN disclosed
US-4716170-A 5-[1H-(5-membered-N-aromatic heteryl)-1-yl]-1,6-naphthyridin-2(1H)-ones and their cardiotonic use STERLING DRUG INC. (US) 1987-12-29 US disclosed
US-4697021-A 1,6-dihydro-6-oxo-3-pyridinecarbonitriles, intermediates for cardiotonic agents STERLING DRUG INC. (US) 1987-09-29 US disclosed
US-4678799-A PARASITICIDES MERCK & CO., INC. (US) 1987-07-07 US disclosed
US-4657915-A INOTROPIC AGENTS STERLING DRUG INC. (US) 1987-04-14 US disclosed
US-4634772-A 2-[2-(di-lower-alkylamino)-1-propenyl]-6-methoxy-3-pyridinecarbonitriles, intermediates for cardiotonic agents STERLING DRUG INC. (US) 1987-01-06 US disclosed
EP-0189853-A2 1,6-Naphthyridin-2(1H)-ones having cardiotonic activity and preparation STERLING DRUG INC. (US) 1986-08-06 EP disclosed
EP-0166533-A1 Quinolone inotropic agents Pfizer Limited (GB) 1986-01-02 EP disclosed
US-4021442-A Production of 1-alkyl-5-nitroimidazoles BASF AKTIENGESELLSCHAFT (DT) 1977-05-03 US disclosed