SCHEMBL7323071

SCHEMBL7323071

Nc1nnc(CCCCN2CC=C(c3ccccc3)CC2)s1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.59
PARP1 P09874 2/20 0.51
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
HTR1A P08908 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
DRD2 P14416 1/20 0.46
TSHR P16473 1/20 0.46
DRD4 P21917 1/20 0.46
CYP2C19 P33261 1/20 0.46
DRD3 P35462 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9138493 0.95 SIGMAR1 (0.53) SIGMAR1PARP1DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL9137258 0.91 L3MBTL1 (0.50) SIGMAR1CYP3A4HTR1ADRD2TSHR
Hydrochloric Acid SCHEMBL9870487 0.80 SIGMAR1 (0.57) SIGMAR1PARP1CYP1A2CYP3A4HTR1A
Hydrochloric Acid SCHEMBL9240174 0.79 SIGMAR1 (0.51) SIGMAR1PARP1HTR1ADRD2
Hydrochloric Acid SCHEMBL9154481 0.79 GRIN2B (0.57) SIGMAR1PARP1HTR1ADRD2DRD4
Hydrochloric Acid SCHEMBL8593986 0.76 GRIN2B (0.55) SIGMAR1CYP3A4HTR1ADRD2TSHR
SCHEMBL7297566 0.76 SIGMAR1 (0.63) SIGMAR1PARP1HTR1ADRD2DRD4
SCHEMBL7270081 0.75 SIGMAR1 (0.51) SIGMAR1PARP1CYP1A2HTR1AMAPT
Hydrochloric Acid SCHEMBL7327180 0.75 SIGMAR1 (0.57) SIGMAR1HTR1ADRD2DRD4DRD3
SCHEMBL10332834 0.74 SIGMAR1 (0.53) SIGMAR1PARP1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0592453-B1 AMINOALKYL-SUBSTITUTED 2-AMINO-1,3,4-THIADIAZOLES, THEIR PREPARATION AND THEIR USE BASF AG (DE) 1998-12-16 EP disclosed
US-5424312-A Treating central nervous system disorders, high blood pressure BASF AKTIENGESELLSCHAFT (DE) 1995-06-13 US disclosed
EP-0592453-A1 AMINOALKYL-SUBSTITUTED 2-AMINO-1,3,4-THIADIAZOLES, THEIR PREPARATION AND THEIR USE BASF Aktiengesellschaft (DE) 1994-04-20 EP disclosed
WO-1992022541-A1 AMINOALKYL-SUBSTITUTED 2-AMINO-1,3,4-THIADIAZOLES, THEIR PREPARATION AND THEIR USE BASF AKTIENGESELLSCHAFT (DE) 1992-12-23 WO disclosed