SCHEMBL7323167

SCHEMBL7323167

NN=Cc1ccc(NC(=O)CCC(=O)NC(CC(=O)O)C(=O)NCCc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.56
ITGA2B P08514 4/20 0.56
POLB P06746 1/20 0.44
KDM1A O60341 1/20 0.43
TSHR P16473 1/20 0.41
CCKBR P32239 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
MDM4 O15151 1/20 0.41
ITGB1 P05556 1/20 0.41
ITGAV P06756 1/20 0.41
ITGA5 P08648 1/20 0.41
MDM2 Q00987 1/20 0.41
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
CA2 P00918 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321045 0.88 ITGB3 (0.44) ITGB3ITGA2BPOLBKDM1ACA2
SCHEMBL7321784 0.85 ITGB3 (0.48) ITGB3ITGA2BCA2
SCHEMBL7331527 0.84 ITGB3 (0.54) ITGB3TSHRITGB1ITGAVITGA5
SCHEMBL7350185 0.84 ITGB3 (0.43) ITGB3ITGA2BPOLBMAPTCA2
SCHEMBL7323153 0.82 ITGB3 (0.65) ITGB3ITGA2B
SCHEMBL8906500 0.82 CA1 (0.46) ITGB3ITGA2BPOLBCA2
SCHEMBL8906494 0.82 CA1 (0.46) ITGB3ITGA2BPOLBCA2
SCHEMBL8895885 0.82 TSHR (0.46) POLBKDM1ATSHRHDAC1HDAC2
SCHEMBL7354349 0.80 ITGB3 (0.67) ITGB3ITGA2B
SCHEMBL7352608 0.78 ITGB3 (0.52) ITGB3ITGA2BPOLBTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5550159-A Peptide mimics useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1996-08-27 US disclosed
US-5453440-A Amidine functional group on benzene ring, anticoagulants G. D. SEARLE & CO. (US) 1995-09-26 US disclosed
WO-1993018058-A1 PEPTIDES MIMICS USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-09-16 WO disclosed