SCHEMBL7323181

SCHEMBL7323181

CCCCN1CCC(CC2C=Cc3c(N)ccc(C(=O)O)c3O2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 14/20 0.48
ADRA2C P18825 3/20 0.41
HTR1D P28221 3/20 0.41
HTR2B P41595 3/20 0.41
HTR3A P46098 3/20 0.41
ADRA1B P35368 2/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM3 P20309 1/20 0.41
ACHE P22303 1/20 0.41
HTR2C P28335 3/20 0.39
ADRA1A P35348 2/20 0.39
ADRA2B P18089 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HTR3D Q70Z44 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7401627 0.78 HTR4 (0.56) HTR4ADRA2CHTR1DHTR2BHTR3A
SCHEMBL8321572 0.72 HTR4 (0.56) HTR4ADRA1BCHRM4CHRM5CHRM3
SCHEMBL4151143 0.71 HTR4 (0.46) HTR4ADRA2CHTR1DHTR2BHTR3A
Hydrochloric Acid SCHEMBL7498481 0.71 HTR4 (0.55) HTR4ADRA1BCHRM4CHRM5CHRM3
SCHEMBL7391971 0.70 HTR4 (0.45) HTR4ADRA2CHTR1DHTR2BHTR3A
SCHEMBL7323178 0.70 HTR4 (0.72) HTR4ADRA2CHTR1DHTR2BHTR3A
Hydrochloric Acid SCHEMBL7417007 0.69 HTR4 (0.46) HTR4ADRA1BCHRM4CHRM5CHRM3
SCHEMBL7411902 0.69 HTR4 (0.46) HTR4ADRA1BCHRM4CHRM5CHRM3
SCHEMBL7405651 0.69 HTR4 (0.55) HTR4ADRA1BCHRM4CHRM5CHRM3
SCHEMBL7401623 0.69 HTR4 (0.52) HTR4ADRA2CHTR1DHTR2BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994008994-A1 HETEROCYCLIC -ESTERS OR -AMIDES USED AS 5-HT4 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-28 WO claimed
US-5708174-A Heterocyclic-esters or -amides used as 5-HT4 receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 1998-01-13 US disclosed
WO-1994008994-A1 HETEROCYCLIC -ESTERS OR -AMIDES USED AS 5-HT4 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-28 WO disclosed