SCHEMBL7323713

SCHEMBL7323713

COc1ccnc(-c2ccc3[nH]cc(C4CCN(C)CC4)c3c2)n1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 0.58
HTR1B P28222 9/20 0.58
HTR1F P30939 5/20 0.58
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
THPO P40225 1/20 0.53
APP P05067 2/20 0.48
HTR1A P08908 3/20 0.47
HTR6 P50406 2/20 0.47
MAPT P10636 1/20 0.46
BLM P54132 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
PIM1 P11309 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
NOS1 P29475 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020706 0.78 HTR1D (0.62) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL8789481 0.76 HTR1D (0.59) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL7710792 0.75 HTR1D (0.67) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL8090606 0.75 KDM4E (0.54) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL8784407 0.75 HTR1D (0.60) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL7014030 0.74 HTR1D (0.57) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL7335724 0.74 HTR6 (0.68) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL7011996 0.74 HTR1F (1.00) HTR1DHTR1BHTR1FHTR1AHTR6
SCHEMBL27498567 0.74 HTR1D (0.66) HTR1DHTR1BHTR1FCYP1A2CYP3A4
SCHEMBL27516181 0.74 HTR1D (0.62) HTR1DHTR1BHTR1FCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed