SCHEMBL7323725

SCHEMBL7323725

CCc1cccc(C)c1OC(CC)(C(=O)O)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
POLB P06746 2/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
MGLL Q99685 1/20 0.38
PTGS2 P35354 1/20 0.38
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
NLRP3 Q96P20 1/20 0.37
PTGER1 P34995 1/20 0.36
PTGER4 P35408 1/20 0.36
PTGER3 P43115 1/20 0.36
PTGER2 P43116 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180298 0.79 KMT2A (0.41) GABRA1GABRB2SMN1; SMN2ALDH1A1TDP1
SCHEMBL16951329 0.75 GABRA1 (0.42) TSHRGABRA1GABRB2SMN1; SMN2ALDH1A1
SCHEMBL982695 0.75 TSHR (0.50) TSHRGABRA1GABRB2SMN1; SMN2ALDH1A1
SCHEMBL7323219 0.74 GABRA1 (0.39) GABRA1GABRB2ALDH1A1TP53KDM4E
SCHEMBL6259721 0.72 PPARA (0.48) TSHRSMN1; SMN2ALDH1A1CYP3A4MGLL
SCHEMBL8166933 0.72 GABRA1 (0.44) TSHRGABRA1GABRB2SMN1; SMN2ALDH1A1
SCHEMBL1805352 0.71 PPARG (0.43) ALDH1A1CYP3A4L3MBTL1KMT2AMAPT
SCHEMBL27641372 0.70 TSHR (0.49) TSHRGABRA1GABRB2SMN1; SMN2ALDH1A1
SCHEMBL13344106 0.70 GABRA1 (0.43) TSHRGABRA1GABRB2SMN1; SMN2ALDH1A1
SCHEMBL16954557 0.69 MAPT (0.44) TSHRGABRA1GABRB2ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526708-B1 Sulfonamide, preparation and use thereof as medicine and intermediate HOFFMANN LA ROCHE (CH) 2000-10-18 EP disclosed
EP-0526708-A1 Sulfonamide, preparation and use thereof as medicine and intermediate F. HOFFMANN-LA ROCHE AG (CH) 1993-02-10 EP disclosed