SCHEMBL7323988

SCHEMBL7323988

NC(C(=O)OCc1ccccc1)C1NC(=O)OC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.46
ALDH1A1 P00352 3/20 0.40
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.39
LTA4H P09960 1/20 0.39
LAP3 P28838 1/20 0.39
KMT2A Q03164 2/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP12 P39900 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013304 0.84 ALDH1A1 (0.43) IDO1ALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL24569694 0.74 CTSD (0.40) ALDH1A1CYP2C9CYP2C19CYP3A4KMT2A
SCHEMBL24569731 0.74 CTSD (0.40) ALDH1A1CYP2C9CYP2C19CYP3A4KMT2A
SCHEMBL9917628 0.73 GLA (0.55) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL9886347 0.73 GLA (0.55) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL4413019 0.73 GLA (0.55) ALDH1A1KMT2AMAPK1L3MBTL1SLC6A2
SCHEMBL21522839 0.72 CYP1A2 (0.42) ALDH1A1SLC1A3SLC1A2SLC1A1CYP1A2
SCHEMBL24569730 0.71 ALDH1A1 (0.39) IDO1ALDH1A1KMT2AMAPK1L3MBTL1
SCHEMBL21274787 0.71 DPP4 (0.55) ALDH1A1CYP2C9CYP2C19CYP3A4LTA4H
SCHEMBL21274786 0.71 DPP4 (0.55) ALDH1A1CYP2C9CYP2C19CYP3A4LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687254-A1 4-AMINOPYRIDINES, THEIR PREPARATION AND THEIR USE AS ANTITHROMBOTIC AGENT Roche Diagnostics GmbH (DE) 1995-12-20 EP disclosed
WO-1994020468-A1 4-AMINOPYRIDINES, THEIR PRODUCTION AND USE AS AN ANTITHROMBOSIS AGENT BOEHRINGER MANNHEIM GMBH (DE) 1994-09-15 WO disclosed
US-4472380-A CARBOXYALKYL DIPEPTIDE DERIVATIVES MERCK & CO., INC. (US) 1984-09-18 US disclosed
US-4374829-A Aminoacid derivatives as antihypertensives MERCK & CO., INC. (US) 1983-02-22 US disclosed
EP-0012401-A1 Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them MERCK & CO. INC. (US) 1980-06-25 EP disclosed