SCHEMBL7324673

SCHEMBL7324673

CCCCN1CCC(CNC(=O)c2cc(Cl)cc3ccoc23)CC1.O=C(O)c1cc(Cl)cc2ccoc12

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.51
HTR4 Q13639 2/20 0.50
CACNA1I Q9P0X4 2/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7331083 0.96 NR4A2 (0.54) NR4A2HTR4CACNA1IKCNH2
SCHEMBL7332743 0.85 HTR4 (0.39) NR4A2HTR4KCNH2
SCHEMBL7332753 0.84 HTR4 (0.53) HTR4
SCHEMBL7324669 0.81 HTR4 (0.38) NR4A2HTR4
SCHEMBL7328044 0.80 HTR4 (0.56) HTR4
SCHEMBL7325370 0.79 NR4A2 (0.54) NR4A2HTR4
SCHEMBL7353765 0.79 NR4A2 (0.51) NR4A2HTR4CACNA1IKCNH2
SCHEMBL7328039 0.76 HTR4 (0.41) NR4A2HTR4KCNH2
SCHEMBL5364372 0.73 HTR4 (0.58) HTR4
SCHEMBL6175694 0.72 NR4A2 (0.49) NR4A2HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664806-A1 HETEROCYCLIC CONDENSED BENZOIC ACID DERIVATIVES AS 5-HT 4? RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-08-02 EP disclosed
WO-1994008995-A1 HETEROCYCLIC CONDENSED BENZOIC ACID DERIVATIVES AS 5-HT4 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-04-28 WO disclosed