SCHEMBL7326381

SCHEMBL7326381

N#Cc1ccc(NC(=O)CCc2ccc(O)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
GAA P10253 1/20 0.58
POLB P06746 3/20 0.56
SAE1 Q9UBE0 1/20 0.55
UBA2 Q9UBT2 1/20 0.55
TRPV1 Q8NER1 1/20 0.55
MAPT P10636 3/20 0.51
CYP1A1 P04798 1/20 0.51
HTT P42858 1/20 0.51
HDAC2 Q92769 3/20 0.51
HDAC8 Q9BY41 3/20 0.51
HDAC3 O15379 2/20 0.51
HDAC4 P56524 2/20 0.51
HDAC1 Q13547 2/20 0.51
HDAC7 Q8WUI4 2/20 0.51
HDAC10 Q969S8 2/20 0.51
HDAC11 Q96DB2 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
HDAC9 Q9UKV0 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29079343 0.85 TRPV1 (0.55) ALDH1A1SMN1; SMN2GAATRPV1MAPT
SCHEMBL3858000 0.83 CNR1 (0.63) ALDH1A1SMN1; SMN2GAAPOLBSAE1
SCHEMBL7302885 0.81 GAA (0.56) ALDH1A1SMN1; SMN2GAAPOLBSAE1
SCHEMBL13776958 0.80 HDAC2 (0.59) SMN1; SMN2GAAPOLBTRPV1MAPT
SCHEMBL19472704 0.80 CNR1 (0.78) SMN1; SMN2POLBSAE1UBA2MAPT
SCHEMBL11705109 0.80 TRPV1 (0.82) SMN1; SMN2GAATRPV1MAPTCYP1A1
SCHEMBL12915848 0.80 MAPT (0.80) ALDH1A1GAATRPV1MAPTCYP1A1
SCHEMBL9261433 0.79 PSMB5 (0.56) ALDH1A1SMN1; SMN2GAAPOLBMAPT
SCHEMBL9268429 0.79 PSMB5 (0.56) ALDH1A1SMN1; SMN2GAAPOLBMAPT
SCHEMBL3084650 0.79 RORC (0.59) ALDH1A1GAAPOLBSAE1UBA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5399585-A Anitcoagulants, antiinflammatory, antitumor HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP disclosed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US disclosed
US-5084466-A Anticoagulants, antiinflammatory agents, atheriosclerosis and antitumor agents HOFFMANN-LA ROCHE INC. (US) 1992-01-28 US disclosed
EP-0381033-A1 Carboxylic-acid and sulphonic-acid amides F. HOFFMANN-LA ROCHE AG (CH) 1990-08-08 EP disclosed