SCHEMBL7326486

SCHEMBL7326486

Cn1c(/C=C/C(=O)O)cc2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.54
ALB P02768 1/20 0.53
PLA2G4A P47712 1/20 0.50
GRIN2D O15399 1/20 0.48
GRIN3B O60391 1/20 0.48
GRIN1 Q05586 1/20 0.48
GRIN2A Q12879 1/20 0.48
GRIN2B Q13224 1/20 0.48
GRIN2C Q14957 1/20 0.48
GRIN3A Q8TCU5 1/20 0.48
DAO P14920 1/20 0.46
KMT2A Q03164 2/20 0.45
PLA2G10 O15496 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SLC9A1 P19634 1/20 0.43
HDAC3 O15379 1/20 0.43
TNKS O95271 1/20 0.43
HDAC4 P56524 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7326492 1.00 MCL1 (0.54) MCL1ALBPLA2G4AGRIN2DGRIN3B
SCHEMBL29247884 0.87 GRIN2D (0.51) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL16756075 0.86 RAB9A (0.51) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL3204520 0.86 ALB (0.49) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL3204531 0.86 ALB (0.49) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL7968178 0.83 MCL1 (0.57) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL6364609 0.83 ALB (0.47) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL6364611 0.83 ALB (0.47) MCL1ALBGRIN2DGRIN3BGRIN1
SCHEMBL19100040 0.80 MCL1 (0.57) MCL1ALBPLA2G4AKMT2AMEN1
SCHEMBL7135266 0.80 TTR (0.45) MCL1ALBGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100495-A4 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORP (US) 2002-09-25 EP disclosed
EP-1100495-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP disclosed
WO-2000006153-A1 PROPENAMIDES AS CCR5 MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed
EP-0392663-A1 Carboline derivative as a 5-HT3 receptor antagonist ONO PHARMACEUTICAL CO., LTD. (JP) 1990-10-17 EP disclosed