SCHEMBL7327316

SCHEMBL7327316

CC[Si](CC)(CC)C(=O)[Si](CC)(CC)CC

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.35
FFAR3 O14843 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6874429 0.74 FFAR3 (0.41) TDP1FFAR3ALDH1A1CES2CES1
SCHEMBL29013295 0.72 ALDH1A1 (0.39) TDP1FFAR3ALDH1A1
SCHEMBL29186273 0.67 ALDH1A1 (0.35) ALDH1A1
SCHEMBL429486 0.65
SCHEMBL30087128 0.65 ALDH1A1 (0.40) TDP1ALDH1A1
SCHEMBL27291347 0.65 ALDH1A1 (0.48) ALDH1A1
SCHEMBL4832765 0.65 FFAR3 (0.33) FFAR3
SCHEMBL149763 0.59 ALDH1A1 (0.41) TDP1FFAR3ALDH1A1CES2CES1
SCHEMBL3230735 0.59 HSD17B10 (0.32) TDP1
Bicarbonate SCHEMBL1127897 0.56 FFAR3 (0.58) TDP1FFAR3ALDH1A1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0378318-A1 Process for synthesis of FK-506 and tricarbonyl intermediates MERCK & CO. INC. (US) 1990-07-18 EP claimed
US-5446158-A Process for synthesis of FK-506 and tricarbonyl intermediates MERCK & CO., INC. (US) 1995-08-29 US disclosed
EP-0378318-A1 Process for synthesis of FK-506 and tricarbonyl intermediates MERCK & CO. INC. (US) 1990-07-18 EP disclosed