SCHEMBL7328394

SCHEMBL7328394

N=C(N)c1ccc(C(=O)NCCCCCNCCC(=O)O)cc1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.63
ITGB3 P05106 17/20 0.56
ITGA2B P08514 17/20 0.56
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14599582 0.87 MAPK1 (0.61) MAPK1ITGB3ITGA2B
SCHEMBL14599618 0.87 MAPK1 (0.61) MAPK1ITGB3ITGA2B
SCHEMBL14599581 0.87 MAPK1 (0.61) MAPK1ITGB3ITGA2B
SCHEMBL14599527 0.87 MAPK1 (0.61) MAPK1ITGB3ITGA2B
SCHEMBL5540645 0.85 MAPK1 (0.58) MAPK1ITGB3ITGA2B
SCHEMBL7304969 0.85 ITGB3 (0.72) MAPK1ITGB3ITGA2B
Hydrochloric Acid SCHEMBL8408094 0.83 MAPK1 (0.68) MAPK1ITGB3ITGA2BCYP1A2CYP2C9
SCHEMBL7306809 0.83 ITGB3 (0.70) MAPK1ITGB3ITGA2B
SCHEMBL8409855 0.83 MAPK1 (0.62) MAPK1ITGB3ITGA2B
SCHEMBL8407980 0.82 F10 (0.60) MAPK1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP claimed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed