SCHEMBL7328407

SCHEMBL7328407

COC(=O)C(O)C(N)CC1CCCCC1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 16/20 0.55
METAP1 P53582 8/20 0.55
REN P00797 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8175196 1.00 METAP2 (0.55) METAP2METAP1REN
Hydrochloric Acid SCHEMBL9514516 0.98 METAP2 (0.53) METAP2METAP1REN
Hydrochloric Acid SCHEMBL9514519 0.98 METAP2 (0.53) METAP2METAP1REN
SCHEMBL8209396 0.95 METAP2 (0.49) METAP2METAP1REN
SCHEMBL13347345 0.95 METAP2 (0.49) METAP2METAP1REN
SCHEMBL8202433 0.95 METAP2 (0.49) METAP2METAP1REN
SCHEMBL13430909 0.91 METAP2 (0.45) METAP2METAP1REN
SCHEMBL10138824 0.91 METAP2 (0.45) METAP2METAP1REN
Trifluoroacetic Acid SCHEMBL7327225 0.90 METAP2 (0.50) METAP2METAP1REN
Hydrochloric Acid SCHEMBL27076653 0.90 METAP2 (0.44) METAP2METAP1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266950-B1 Nor-statine and nor-cyclostatine polypeptides PFIZER (US) 1993-12-29 EP disclosed
US-5095119-A Renin inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1992-03-10 US disclosed
US-5075451-A Pyrrolimidazolones useful as renin inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1991-12-24 US disclosed
US-5064965-A Renin inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1991-11-12 US disclosed
US-5034376-A Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1991-07-23 US disclosed
US-5023338-A Renin inhibitors AMERICAN HOME PRODUCTS CORPORATION (US) 1991-06-11 US disclosed
EP-0266950-A2 Nor-statine and nor-cyclostatine polypeptides PFIZER INC. (US) 1988-05-11 EP disclosed