SCHEMBL8202433

SCHEMBL8202433

COC(=O)C(O)C(N)CC1CCC1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 17/20 0.49
METAP1 P53582 8/20 0.49
REN P00797 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13347345 1.00 METAP2 (0.49) METAP2METAP1REN
SCHEMBL8209396 1.00 METAP2 (0.49) METAP2METAP1REN
SCHEMBL7328407 0.95 METAP2 (0.55) METAP2METAP1REN
SCHEMBL8175196 0.95 METAP2 (0.55) METAP2METAP1REN
Hydrochloric Acid SCHEMBL9514519 0.93 METAP2 (0.53) METAP2METAP1REN
Hydrochloric Acid SCHEMBL9514516 0.93 METAP2 (0.53) METAP2METAP1REN
SCHEMBL10138824 0.93 METAP2 (0.45) METAP2METAP1REN
SCHEMBL13430909 0.93 METAP2 (0.45) METAP2METAP1REN
Hydrochloric Acid SCHEMBL27076653 0.91 METAP2 (0.44) METAP2METAP1REN
Trifluoroacetic Acid SCHEMBL7327225 0.85 METAP2 (0.50) METAP2METAP1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104292130-B A kind of synthetic method of EBP520 intermediate 2-hydroxyl-3-amino-4-cyclobutyl butanamide hydrochloride SUZHOU UUGENE BIOPHARMA CO., LTD. (CN) 2016-04-27 CN claimed
CN-104292130-B A kind of synthetic method of EBP520 intermediate 2-hydroxyl-3-amino-4-cyclobutyl butanamide hydrochloride SUZHOU UUGENE BIOPHARMA CO., LTD. (CN) 2016-04-27 CN disclosed
US-RE43298-E1 Peptides as NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2012-04-03 US disclosed
EP-1730142-B1 NOVEL KETOAMIDES WITH CYCLIC P4'S AS INHIBITORS OF NS3 SERINE PROTEASE OF HEPATITIS C VIRUS SCHERING CORP (US) 2011-06-29 EP disclosed
EP-1939213-B1 Novel compounds as inhibitors of hepatitis C virus NS3 serine protease SCHERING CORP (US) 2010-08-25 EP disclosed
US-7759499-B2 Compounds as inhibitors of hepatitis C virus NS3 serine protease SCHERING CORPORATION (US) 2010-07-20 US disclosed
EP-1730110-B1 SULFUR COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORP (US) 2010-06-09 EP disclosed
US-20100113821-A1 PREPARATION OF 3-AMINO-3-(CYCLOBUTYLMETHYL)-2-(HYDROXY)-PROPIONAMIDE HYDROCHLORIDE SCHERING-PLOUGH CORPORATION (US) 2010-05-06 US disclosed
US-20100113821-A1 PREPARATION OF 3-AMINO-3-(CYCLOBUTYLMETHYL)-2-(HYDROXY)-PROPIONAMIDE HYDROCHLORIDE SCHERING-PLOUGH CORPORATION (US) 2010-05-06 US disclosed
EP-1385870-B1 PEPTIDES AS NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS SCHERING CORP (US) 2010-03-17 EP disclosed
WO-2006130686-A2 HCV PROTEASE INHIBITORS IN COMBINATION WITH FOOD SCHERING CORPORATION (US) 2006-12-07 WO disclosed
WO-2005113581-A1 SUBSTITUTED PROLINES AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-12-01 WO disclosed
WO-2005107745-A1 AN INHIBITOR OF HEPATITIS C SCHERING CORPORATION (US) 2005-11-17 WO disclosed
WO-2005087730-A1 3,4-(CYCLOPENTYL)-FUSED PROLINE COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-09-22 WO disclosed
WO-2005087721-A2 COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-09-22 WO disclosed
WO-2005087725-A2 NOVEL COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-09-22 WO disclosed
WO-2005087731-A1 SULFUR COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-09-22 WO disclosed
WO-2005085242-A1 NOVEL KETOAMIDES WITH CYCLIC P4'S AS INHIBITORS OF NS3 SERINE PROTEASE OF HEPATITIS C VIRUS SCHERING CORPORATION (US) 2005-09-15 WO disclosed
WO-2005085275-A1 INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE SCHERING CORPORATION (US) 2005-09-15 WO disclosed
WO-2003062265-A2 NOVEL PEPTIDES AS NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS SCHERING CORPORATION (US) 2003-07-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113821-A1 PREPARATION OF 3-AMINO-3-(CYCLOBUTYLMETHYL)-2-(HYDROXY)-PROPIONAMIDE HYDROCHLORIDE CTRL, DNPEP, DPP3 METAP2 144/4885METAP1 29/4885REN 669/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.