SCHEMBL7328837

SCHEMBL7328837

c1ccc(C(N=C2CCCCCCCN2)c2ccccc2)cc1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A2 P05177 3/20 0.32
CYP3A4 P08684 3/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
KCNA5 P22460 2/20 0.32
CYP2C19 P33261 2/20 0.32
KCNH2 Q12809 2/20 0.32
KCNE1 P15382 1/20 0.32
NISCH Q9Y2I1 1/20 0.30
KDM4E B2RXH2 3/20 0.30
MEN1 O00255 3/20 0.30
KMT2A Q03164 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327602 1.00 NPC1 (0.33) NPC1HPGDRAB9ASMN1; SMN2CYP1A2
SCHEMBL7325279 1.00 NPC1 (0.33) NPC1HPGDRAB9ASMN1; SMN2CYP1A2
SCHEMBL7325274 1.00 NPC1 (0.33) NPC1HPGDRAB9ASMN1; SMN2CYP1A2
SCHEMBL7327606 1.00 NPC1 (0.33) NPC1HPGDRAB9ASMN1; SMN2CYP1A2
SCHEMBL11875818 0.91 HTR2A (0.36) MEN1KMT2A
SCHEMBL7327733 0.91 SLC6A2 (0.36) HPGDSMN1; SMN2CYP1A2CYP3A4CYP2D6
SCHEMBL7336045 0.91 HTR2A (0.36) MEN1KMT2A
Hydrochloric Acid SCHEMBL11872449 0.91 CHRNB2 (0.33) NPC1HPGDSMN1; SMN2CYP3A4KCNH2
SCHEMBL7336042 0.91 HTR2A (0.36) MEN1KMT2A
Hydrochloric Acid SCHEMBL11879426 0.90 HTR2A (0.35) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198433-A Hypotensive MERRELL DOW PHARMACEUTICALS INC. (US) 1993-03-30 US disclosed
US-5158945-A Cardiotonic agents, vasodilators, hypotensive agents, anticonvulsants, antiisichemic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-10-27 US disclosed
EP-0370320-B1 LACTAMIMIDES IN THE TREATMENT OF DRUG-RESISTANT PROTOZOAL INFECTIONS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-09-30 EP disclosed
US-5128337-A Hypotensive agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-07-07 US disclosed
US-5082837-A Hypotensive MERRELL DOW PHARMACEUTICALS (US) 1992-01-21 US disclosed
US-5010072-A Hypotensive agents MERRELL DOW PHARMACEUTICALS INC. (US) 1991-04-23 US disclosed
EP-0370320-A1 Lactamimides in the treatment of drug-resistant protozoal infections MERRELL DOW PHARMACEUTICALS INC. (US) 1990-05-30 EP disclosed
EP-0348891-A2 Lactamimides as calcium antagonists MERRELL DOW PHARMACEUTICALS INC. (US) 1990-01-03 EP disclosed
US-4061746-A Lactamimide inhibitors of gastrointestinal hypersecretion RICHARDSON-MERRELL INC. (US) 1977-12-06 US disclosed