SCHEMBL7329018

SCHEMBL7329018

CCc1cccc(CN(C)C(=O)N[C@H](C(=O)O)C(C)C)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.47
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
PDE5A O76074 1/20 0.40
MME P08473 1/20 0.40
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
EGLN1 Q9GZT9 2/20 0.37
PPARG P37231 2/20 0.37
PPARA Q07869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329148 1.00 CA2 (0.47) CA2ALDH1A1POLBPDE5AMME
SCHEMBL7308687 0.87 CA2 (0.47) CA2ALDH1A1POLBMMEGAA
SCHEMBL7308684 0.87 CA2 (0.47) CA2ALDH1A1POLBMMEGAA
SCHEMBL4683895 0.81 CA2 (0.67) CA2ALDH1A1POLBMMEGAA
SCHEMBL4683897 0.81 CA2 (0.67) CA2ALDH1A1POLBMMEGAA
SCHEMBL7337373 0.80 CYP1A2 (0.48) CA2ALDH1A1GAANPSR1CYP1A2
SCHEMBL7337376 0.80 CYP1A2 (0.48) CA2ALDH1A1GAANPSR1CYP1A2
SCHEMBL1058928 0.79 PDE5A (0.41) CA2ALDH1A1PDE5ACYP2C19
SCHEMBL7094675 0.78 CYP3A4 (0.42) CA2CYP3A4CYP1A2CYP2D6CYP2C19
SCHEMBL5711217 0.76 NPC1 (0.56) CA2ALDH1A1POLBGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990135-A FOR TREATING A RETROVIRAL INFECTION SUCH AS HIV INFECTION; FOR EXAMPLE 5S-N-((2-PYRIDINYL)METHOXYCARBONYL)VALINYLAMINO-2-((N-3 -PYRIDINYL)METHOXYCARBONYL)AMINO-4S-HYDROXY-1,6-DIPHENYL-2-AZAHEXANE AND OTHER COMPOUNDS OF GIVEN FORMULA ABBOTT LABORATORIES (US) 1999-11-23 US disclosed
US-5631376-A PEPTIDE DERIVATIVES FOR TREATMENT OF AIDS ABBOTT LABORATORIES (US) 1997-05-20 US disclosed
US-5621109-A OXAZOLE/THIAZOLE DERIVATIVES OF HYDROXYMETHYL HYDRAZONES; SIDE EFFECT REDUCTION ABBOTT LABORATORIES (US) 1997-04-15 US disclosed
EP-0683772-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1995-11-29 EP disclosed
US-5461067-A For HIV infections ABBOTT LABORATORIES (US) 1995-10-24 US disclosed
EP-0683772-A4 RETROVIRAL PROTEASE INHIBITING COMPOUNDS. ABBOTT LAB (US) 1995-09-27 EP disclosed
WO-1994019332-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1994-09-01 WO disclosed