SCHEMBL7337376

SCHEMBL7337376

CC(C)[C@H](NC(=O)N(C)Cc1ccc2ccccc2n1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
ADAMTS4 O75173 2/20 0.48
CA2 P00918 2/20 0.45
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
PRNP P04156 1/20 0.44
MAPK10 P53779 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
AGTR2 P50052 1/20 0.42
PDK1 Q15118 1/20 0.41
PDE10A Q9Y233 4/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337373 1.00 CYP1A2 (0.48) CYP1A2ADAMTS4CA2ALDH1A1KDM4E
SCHEMBL27372584 0.91 CYP1A2 (0.44) CYP1A2ADAMTS4CA2ALDH1A1KDM4E
SCHEMBL7305142 0.91 CYP1A2 (0.44) CYP1A2ADAMTS4CA2ALDH1A1KDM4E
SCHEMBL7388688 0.89 CYP1A2 (0.43) CYP1A2ADAMTS4CA2ALDH1A1KDM4E
SCHEMBL27375082 0.84 HDAC1 (0.46) CYP1A2ALDH1A1KDM4EPRNPMAPK10
SCHEMBL7300357 0.84 HDAC1 (0.46) CYP1A2ALDH1A1KDM4EPRNPMAPK10
SCHEMBL7298672 0.83 CYP1A2 (0.43) CYP1A2ALDH1A1KDM4EPRNPMAPK10
SCHEMBL7300431 0.81 MME (0.44) CYP1A2ALDH1A1HDAC1HDAC2AGTR2
SCHEMBL7329343 0.81 CYP1A2 (0.41) CYP1A2ADAMTS4ALDH1A1KDM4EPRNP
SCHEMBL7329018 0.80 CA2 (0.47) CYP1A2CA2ALDH1A1NPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed