SCHEMBL732923

SCHEMBL732923

Nc1ccc(O)c(C(=O)NO)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.64
KDM4E B2RXH2 4/20 0.62
TDP1 Q9NUW8 3/20 0.62
HIF1A Q16665 2/20 0.62
ALDH1A1 P00352 2/20 0.62
CYP3A4 P08684 2/20 0.62
MEN1 O00255 2/20 0.62
THRB P10828 2/20 0.62
RECQL P46063 2/20 0.62
KMT2A Q03164 2/20 0.62
ALOX15 P16050 2/20 0.62
HSD17B10 Q99714 2/20 0.62
TNF P01375 1/20 0.62
HSPD1 P10809 1/20 0.62
CYP2C9 P11712 1/20 0.62
HPGD P15428 1/20 0.62
CASP1 P29466 1/20 0.62
CYP2C19 P33261 1/20 0.62
PTGS2 P35354 1/20 0.62
KDR P35968 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1555835 0.84 KDM4E (0.62) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL2299271 0.82 ALOX5 (0.67) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL14215697 0.82 MAPT (0.59) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL17774881 0.79 P2RX1 (0.60) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL15894582 0.79 ALOX5 (0.63) ALOX5KDM4ETDP1HIF1AALDH1A1
Mesalamine SCHEMBL28187698 0.79 KDM4E (0.96) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL9312494 0.79 EGFR (0.61) ALOX5KDM4EHIF1AALDH1A1PTGS2
SCHEMBL16589373 0.78 CASP1 (0.45) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL1977469 0.78 ALOX5 (0.61) ALOX5KDM4ETDP1HIF1AALDH1A1
SCHEMBL9363663 0.78 ALOX5 (1.00) ALOX5KDM4ETDP1HIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116602950-A Methods of treating fibrosis 诺格拉制药有限公司 2023-08-18 CN disclosed
WO-2020056044-A1 MODIFIED ARCHAEAL FAMILY B POLYMERASES Singular Genomics Systems, Inc. (US) 2020-03-19 WO disclosed
US-8450506-B2 Compounds and their salts specific to the PPAR receptors and the EGF Receptors and their use in the medical field NOGRA PHARMA LIMITED (IE) 2013-05-28 US disclosed
US-8450506-B2 Compounds and their salts specific to the PPAR receptors and the EGF Receptors and their use in the medical field NOGRA PHARMA LIMITED (IE) 2013-05-28 US disclosed
US-20120316230-A1 Compounds and their Salts Specific to the PPAR Receptors and the EGF Receptors and their Use in the Medical Field GIULIANI INTERNATIONAL LIMITED (IE) 2012-12-13 US disclosed
US-20120316230-A1 Compounds and their Salts Specific to the PPAR Receptors and the EGF Receptors and their Use in the Medical Field GIULIANI INTERNATIONAL LIMITED (IE) 2012-12-13 US disclosed
US-8138357-B2 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field GIULIANI INTERNATIONAL LIMITED (IE) 2012-03-20 US disclosed
US-8138357-B2 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field GIULIANI INTERNATIONAL LIMITED (IE) 2012-03-20 US disclosed
US-20110152225-A1 PPAR-Gamma Agonists for the Induction of Cationic Antimicrobial Peptide Expression as Immunoprotective Stimulants NOGRA PHARMA LIMITED (IE) 2011-06-23 US disclosed
US-20110152225-A1 PPAR-Gamma Agonists for the Induction of Cationic Antimicrobial Peptide Expression as Immunoprotective Stimulants NOGRA PHARMA LIMITED (IE) 2011-06-23 US disclosed
US-20090118357-A1 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field GIULIANI INTERNATIONAL LIMITED (IE) 2009-05-07 US disclosed
US-20090118357-A1 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field GIULIANI INTERNATIONAL LIMITED (IE) 2009-05-07 US disclosed
US-20030171260-A1 Compositions and methods utilizing hydroxamates to scavenge oxidant toxins NELSON DEANNA JEAN (US) 2003-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090118357-A1 Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field EGFR, ERBB3, FGFR3 ALOX5 2705/4885KDM4E 4603/4885TDP1 4868/4885
US-20120316230-A1 Compounds and their Salts Specific to the PPAR Receptors and the EGF Receptors and their Use in the Medical Field EGFR, ERBB3, FGFR3 ALOX5 2274/4885KDM4E 4435/4885TDP1 4867/4885
US-20110152225-A1 PPAR-Gamma Agonists for the Induction of Cationic Antimicrobial Peptide Expression as Immunoprotective Stimulants PPARG, FABP2, PPARD ALOX5 428/4885KDM4E 4571/4885TDP1 3605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.