SCHEMBL7330868

SCHEMBL7330868

CC(C)(C)OC(=O)N1C(=O)CC(=O)[C@H]1CC1CCCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
BACE1 P56817 2/20 0.35
HPGD P15428 1/20 0.35
CTSD P07339 1/20 0.35
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
NR1H2 P55055 1/20 0.33
GLS O94925 1/20 0.32
KLK7 P49862 1/20 0.32
GAA P10253 1/20 0.32
FEN1 P39748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29526186 0.93 NR1H2 (0.38) CHRM2CHRM1CHRM3HPGDDDB1
SCHEMBL20734866 0.77 KLK7 (0.36) CHRM2CHRM1CHRM3DDB1CRBN
SCHEMBL20734867 0.77 KLK7 (0.36) CHRM2CHRM1CHRM3DDB1CRBN
SCHEMBL32683207 0.77 CHRM2 (0.35) CHRM2CHRM1CHRM3CTSKDDB1
SCHEMBL7340433 0.76 CHRM2 (0.41) EPHX1CHRM2CHRM1CHRM3BACE1
SCHEMBL5963373 0.75 EPHX1 (0.37) EPHX1CHRM2CHRM1CHRM3BACE1
SCHEMBL20734946 0.75 CHRM2 (0.33) CHRM2CHRM1CHRM3DDB1CRBN
SCHEMBL20734945 0.75 CHRM2 (0.33) CHRM2CHRM1CHRM3DDB1CRBN
SCHEMBL2196268 0.73 CHRM2 (0.41) CHRM2CHRM1CHRM3HPGDDDB1
SCHEMBL2196261 0.73 CHRM2 (0.41) CHRM2CHRM1CHRM3HPGDDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed