SCHEMBL5963373

SCHEMBL5963373

CC(C)(C)OC(=O)N1C(=O)[C@H](O)[C@@H]1CC1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
HPGD P15428 1/20 0.36
BACE1 P56817 2/20 0.36
CTSD P07339 1/20 0.36
NR1H2 P55055 1/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
GLS O94925 1/20 0.33
NAAA Q02083 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340433 0.83 CHRM2 (0.41) EPHX1CHRM2CHRM1CHRM3HPGD
SCHEMBL7339735 0.78 KLK7 (0.43) KMT2APDE4APDE4BPDE4CPDE4D
SCHEMBL5963853 0.77 BACE1 (0.31) EPHX1HPGDBACE1CTSDALDH1A1
SCHEMBL5964671 0.76 EPHX1 (0.40) EPHX1CHRM2CHRM1CHRM3HPGD
SCHEMBL5964675 0.76 EPHX1 (0.40) EPHX1CHRM2CHRM1CHRM3HPGD
SCHEMBL5963617 0.76 KLK7 (0.36) CHRM2CHRM1CHRM3NR1H2ALDH1A1
SCHEMBL7979086 0.76 KLK7 (0.36) CHRM2CHRM1CHRM3NR1H2ALDH1A1
SCHEMBL7330868 0.75 EPHX1 (0.36) EPHX1CHRM2CHRM1CHRM3HPGD
SCHEMBL31735232 0.71 NR1H2 (0.53) EPHX1HPGDBACE1CTSDNR1H2
SCHEMBL19217730 0.71 EPHX1 (0.46) EPHX1CHRM2CHRM1CHRM3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0681568-B1 PROCESS FOR PREPARATION OF TAXANE DERIVATIVES AND BETA-LACTAM INTERMEDIATES THEREFOR UNIV NEW YORK STATE RES FOUND (US) 2006-07-26 EP disclosed
US-6218553-B1 METALLIZATION BY REACTING A BACCATIN III DERIVATIVE WITH A METAL ALKYLDISILAZIDE THE STATE UNIVERSITY OF NEW YORK AT STONY BROOK 2001-04-17 US disclosed
US-6187916-B1 Process for the preparation of taxane derivatives and β-lactam intermediates therefor RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK 2001-02-13 US disclosed