SCHEMBL7333545

SCHEMBL7333545

CC(C)[C@H](NC(=O)CCc1nccs1)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)CCc1nccs1)C(C)C

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.54
CTSD P07339 9/20 0.45
PKM P14618 1/20 0.42
HSPA5 P11021 1/20 0.42
HSPA9 P38646 1/20 0.42
BACE1 P56817 1/20 0.42
REN P00797 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7341787 0.98 CA2 (0.52) CA2CTSDPKMHSPA5HSPA9
SCHEMBL7338391 0.89 CA2 (0.58) CA2CTSDBACE1REN
SCHEMBL7339220 0.83 CA2 (0.71) CA2CTSDHSPA5HSPA9BACE1
SCHEMBL7339544 0.83 CA2 (0.71) CA2CTSDHSPA5HSPA9BACE1
SCHEMBL7339662 0.83 CA2 (0.71) CA2CTSDHSPA5HSPA9BACE1
SCHEMBL6449601 0.83 CA2 (0.70) CA2CTSD
SCHEMBL7269664 0.82 CTSD (0.58) CA2CTSD
SCHEMBL6447523 0.81 CA2 (0.54) CA2CTSDBACE1REN
SCHEMBL7269412 0.81 CA2 (0.67) CA2CTSD
SCHEMBL7330968 0.79 CA2 (0.65) CA2CTSDHSPA5HSPA9BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed