SCHEMBL7334346

SCHEMBL7334346

COCCCCCOc1ccc(-c2ccc(B(O)O)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
RARB P10826 4/20 0.45
HDAC3 O15379 6/20 0.44
HDAC4 P56524 6/20 0.44
HDAC1 Q13547 6/20 0.44
HDAC7 Q8WUI4 6/20 0.44
HDAC2 Q92769 6/20 0.44
HDAC10 Q969S8 6/20 0.44
HDAC11 Q96DB2 6/20 0.44
HDAC8 Q9BY41 6/20 0.44
HDAC6 Q9UBN7 6/20 0.44
HDAC9 Q9UKV0 6/20 0.44
HDAC5 Q9UQL6 6/20 0.44
GAA P10253 1/20 0.42
NR5A1 Q13285 1/20 0.42
MGLL Q99685 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7334085 1.00 ENPP2 (0.48) ENPP2CA1CA2RARBHDAC3
SCHEMBL2561437 0.90 CA2 (0.55) ENPP2CA1CA2GAANR5A1
SCHEMBL7698504 0.87 RARB (0.60) CA1CA2RARBGAANR5A1
SCHEMBL1792038 0.87 RARB (0.60) CA1CA2RARBGAANR5A1
SCHEMBL5392482 0.87 RARB (0.60) CA1CA2RARBGAANR5A1
SCHEMBL3039053 0.87 RARB (0.60) CA1CA2RARBGAANR5A1
SCHEMBL20312081 0.86 CYP3A4 (0.52) RARBHDAC3HDAC4HDAC1HDAC7
SCHEMBL2555796 0.85 RARB (0.58) CA1CA2RARBNR5A1MGLL
SCHEMBL3036082 0.84 CYP2D6 (0.58) ENPP2CA1CA2RARBNR5A1
SCHEMBL247173 0.84 CA2 (0.57) ENPP2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0854140-B1 Vitronectin receptor antagonists, their production and their use SANOFI AVENTIS DEUTSCHLAND (DE) 2013-11-06 EP disclosed
EP-0788511-B1 CYCLIC HEXAPEPTIDES HAVING ANTIBIOTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO (JP) 2002-12-11 EP disclosed
US-6265536-B1 MICROBIOCIDE AND FUNGICIDE WHICH IS INHIBITOR OF BETA-1,3-GLUCAN SYNTHASE; TREATMENT OF PNEUMOCYSTIS CARINII INFECTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-07-24 US disclosed
US-6107458-A FUNGICIDE WHICH IS BETA-1,3-GLYCAN SYNTHASE INHIBITOR; FOR PROPHYLAXIS AND TREATMENT OF PNEUMOCYSTIS CARINII INFECTIONS LIKE PNEUMONIA FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-08-22 US disclosed
EP-0854140-A2 Vitronectin receptor antagonists, their production and their use HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-22 EP disclosed
EP-0788511-A1 CYCLIC HEXAPEPTIDES HAVING ANTIBIOTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-08-13 EP disclosed
WO-1996011210-A1 CYCLIC HEXAPEPTIDES HAVING ANTIBIOTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-04-18 WO disclosed