SCHEMBL7336199

SCHEMBL7336199

CC(I)c1cccc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.53
HTR2A P28223 3/20 0.50
HTR2B P41595 3/20 0.50
HTR2C P28335 2/20 0.50
IDO1 P14902 1/20 0.50
TDO2 P48775 1/20 0.50
DAO P14920 1/20 0.50
ACP3 P15309 2/20 0.49
CES2 O00748 2/20 0.49
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.45
SLC6A4 P31645 2/20 0.44
SIGMAR1 Q99720 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
ADRA2C P18825 1/20 0.44
ADRA1A P35348 1/20 0.44
DRD3 P35462 1/20 0.44
OPRK1 P41145 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23343776 1.00 PNMT (0.53) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL2601113 0.85 DAO (0.59) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL255035 0.85 PNMT (0.55) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL15820267 0.83 HTR2A (0.51) PNMTHTR2AHTR2BHTR2CIDO1
Ammonia Solution, Strong SCHEMBL27629775 0.83 PNMT (0.53) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL22189207 0.83 PNMT (0.56) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL215226 0.82 PNMT (0.51) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL1535283 0.82 PNMT (0.61) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL22497538 0.82 PNMT (0.51) PNMTHTR2AHTR2BHTR2CIDO1
SCHEMBL10157207 0.82 PNMT (0.51) PNMTHTR2AHTR2BHTR2CIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2650286-A1 Quinazoline derivatives and therapeutic use thereof Rexahn Pharmaceuticals, Inc. (US) 2013-10-16 EP disclosed
EP-0771196-A4 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 1997-09-03 EP disclosed
EP-0771196-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-05-07 EP disclosed
WO-1996007405-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-03-14 WO disclosed