SCHEMBL7336648

SCHEMBL7336648

Cc1c([N+](=O)[O-])ccc(OS(=O)(=O)C(F)(F)F)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
EPAS1 Q99814 3/20 0.39
TDP1 Q9NUW8 5/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
TTR P02766 2/20 0.38
ALB P02768 1/20 0.38
THRB P10828 1/20 0.38
PTPN1 P18031 1/20 0.38
TSHR P16473 3/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
HIF1A Q16665 1/20 0.36
TXNRD1 Q16881 1/20 0.36
TXNRD3 Q86VQ6 1/20 0.36
TXNRD2 Q9NNW7 1/20 0.36
PPOX P50336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4471027 0.87 TDP1 (0.41) CRHBPCRHR2EPAS1TDP1MEN1
SCHEMBL7550828 0.80 TSHR (0.49) MEN1KMT2APTPN1TSHRALDH1A1
SCHEMBL4003073 0.78 EPAS1 (0.41) EPAS1TDP1MEN1KMT2ATTR
SCHEMBL31090845 0.77 PDE7A (0.49) EPAS1KMT2APTPN1TSHRALDH1A1
SCHEMBL6816625 0.77 PDE7A (0.49) EPAS1KMT2APTPN1TSHRALDH1A1
SCHEMBL810810 0.77 TSHR (0.49) TDP1MEN1KMT2APTPN1TSHR
SCHEMBL31090816 0.77 TSHR (0.49) TDP1MEN1KMT2APTPN1TSHR
SCHEMBL7392580 0.77 TSHR (0.40) CRHBPCRHR2TDP1MEN1KMT2A
SCHEMBL2050119 0.77 TDP1 (0.39) CRHBPCRHR2EPAS1TDP1THRB
SCHEMBL8548365 0.76 TDP1 (0.50) TDP1MEN1KMT2ATTRALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674620-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014771-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed