SCHEMBL7337104

SCHEMBL7337104

COc1ccc(-c2c(-c3ccccc3)ccc(S(N)(=O)=O)c2-c2onc(C)c2Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 4/20 0.43
EDNRA P25101 4/20 0.43
BRD4 O60885 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
S1PR1 P21453 1/20 0.38
NR1H4 Q96RI1 1/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 1/20 0.38
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP3A4 P08684 2/20 0.37
PTGS2 P35354 2/20 0.37
MT-CO2 P00403 1/20 0.37
CA3 P07451 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6151087 0.82 CA2 (0.48) EDNRBEDNRALMNACA12CA1
SCHEMBL27474879 0.81 EDNRB (0.43) EDNRBEDNRABRD4NR1H4LMNA
SCHEMBL7337110 0.80 CA2 (0.46) EDNRBEDNRALMNACA12CA1
SCHEMBL6151278 0.79 PTGS2 (0.47) EDNRBEDNRALMNACA12CA1
SCHEMBL7337092 0.77 CA2 (0.44) EDNRBEDNRASMN1; SMN2NR1H4LMNA
SCHEMBL27492675 0.77 CA2 (0.44) EDNRBEDNRASMN1; SMN2NR1H4CA12
SCHEMBL6151358 0.77 CA2 (0.47) EDNRBEDNRALMNACA12CA1
SCHEMBL6151081 0.76 PTGS2 (0.51) EDNRBEDNRALMNACA12CA1
SCHEMBL7211619 0.75 PTGS2 (0.46) EDNRBEDNRALMNACA12CA1
SCHEMBL27454564 0.73 CA2 (0.56) EDNRBEDNRABRD4CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819125-A1 THIENYL-, FURYL-, PYRROLYL- AND BIPHENYLSULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1998-01-21 EP disclosed
WO-1996031492-A1 THIENYL-, FURYL-, PYRROLYL- AND BIPHENYLSULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-10-10 WO disclosed