SCHEMBL7337295

SCHEMBL7337295

CC(C[CH]C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)Nc1nccs1)C(N)=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPA5 P11021 4/20 0.54
HSPA2 P54652 2/20 0.54
HSPA1A P0DMV8 1/20 0.54
HSPA9 P38646 1/20 0.54
PKM P14618 1/20 0.47
PPARG P37231 3/20 0.46
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ITGA4 P13612 1/20 0.43
MME P08473 1/20 0.43
ACE P12821 1/20 0.43
CPA1 P15085 1/20 0.43
ACE2 Q9BYF1 1/20 0.43
PIN1 Q13526 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
LMNA P02545 2/20 0.43
XBP1 P17861 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7025425 0.92 HSPA5 (0.63) HSPA5HSPA2HSPA1AHSPA9PKM
SCHEMBL7344073 0.84 PPARG (0.62) PPARGMMP9MMP8MMEACE
SCHEMBL7344259 0.84 MEN1 (0.52) PPARGMMP9MMP8MMEACE
SCHEMBL7348738 0.83 NPC1 (0.54) PPARGMMP9MMP8HDAC6MME
SCHEMBL7336531 0.83 NPC1 (0.54) PPARGMMP9MMP8HDAC6MME
SCHEMBL7342788 0.83 NPC1 (0.54) PPARGMMP9MMP8HDAC6MME
SCHEMBL7345065 0.83 HDAC8 (0.56) PPARGMMP9MMP8HDAC6MME
SCHEMBL7338315 0.83 PPARG (0.52) PPARGMMP9MMP8MMEACE
SCHEMBL7337025 0.83 KLKB1 (0.52) PPARGMMP9MMP8MMEACE
SCHEMBL7338154 0.82 PPARG (0.51) PPARGMMP9MMP8MMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US claimed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed