SCHEMBL7337339

SCHEMBL7337339

COC(=O)C1=C(O)c2cc3c(cc2S(=O)(=O)N1)OCO3

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 2/20 0.36
TSHR P16473 1/20 0.36
PTGES O14684 3/20 0.36
KDM4E B2RXH2 4/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.35
ATM Q13315 1/20 0.35
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
NR4A1 P22736 1/20 0.34
RECQL P46063 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337154 0.79 PTGES (0.47) KMT2AMAPTPTGESKDM4E
SCHEMBL7336011 0.75 SMN1; SMN2 (0.41) SMN1; SMN2MEN1KMT2AALDH1A1MAPT
SCHEMBL11490983 0.75 PTGES (0.47) PTGES
SCHEMBL11493406 0.75 PTGES (0.47) ALDH1A1PTGESKDM4E
SCHEMBL7337108 0.74 PTGES (0.59) ALDH1A1MAPTPTGESKDM4E
SCHEMBL11487687 0.74 CHEK1 (0.54) PTGES
SCHEMBL7342661 0.72 PTGES (0.56) KMT2APTGESKDM4E
SCHEMBL30940077 0.72 PTGES (0.56) KMT2APTGESKDM4E
SCHEMBL8799145 0.72 TARBP2 (0.31)
SCHEMBL7336002 0.66 SMN1; SMN2 (0.47) SMN1; SMN2MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811001-B1 BENZOTHIAZINE DIOXIDES AS ENDOTHELIN ANTAGONISTS WARNER LAMBERT CO (US) 2001-10-31 EP disclosed
WO-1996026195-A1 BENZOTHIAZINE DIOXIDES AS ENDOTHELIN ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1996-08-29 WO disclosed