SCHEMBL7338355

SCHEMBL7338355

CC(C)[C@H](NC(=O)N1CCN(C)CC1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)N1CCN(C)CC1)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.52
HSD17B10 Q99714 1/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CTSS P25774 2/20 0.48
CTSL P07711 2/20 0.48
CHRM1 P11229 2/20 0.47
CTSD P07339 2/20 0.47
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CTSB P07858 2/20 0.45
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343714 0.91 CTSD (0.61) CA2MEN1KMT2ACTSSCTSL
SCHEMBL7336891 0.91 KLK5 (0.52) KMT2ACTSD
SCHEMBL7339472 0.90 CYP2C19 (0.58) CA2MEN1KMT2ACTSSCTSD
SCHEMBL7333266 0.90 CYP2C19 (0.58) CA2MEN1KMT2ACTSSCTSD
SCHEMBL7335199 0.90 CYP2C19 (0.58) CA2MEN1KMT2ACTSSCTSD
SCHEMBL7280132 0.89 CTSD (0.61) MEN1KMT2ACTSSCTSLCTSD
SCHEMBL7333752 0.89 POLB (0.58) CA2HSD17B10MEN1KMT2ACTSS
SCHEMBL7333759 0.89 POLB (0.58) CA2HSD17B10MEN1KMT2ACTSS
SCHEMBL7301749 0.89 POLB (0.58) CA2HSD17B10MEN1KMT2ACTSS
SCHEMBL7337580 0.85 CA2 (0.79) CA2HSD17B10MEN1KMT2ACTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5914319-A Antithrombotic agents ELI LILLY AND COMPANY (US) 1999-06-22 US disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5726159-A PEPTIDE THROMBIN INHIBITORS ELI LILLY AND COMPANY (US) 1998-03-10 US disclosed
US-5710130-A HETEROCYCLIC SYNTHETIC PEPTIDES ELI LILLY AND COMPANY (US) 1998-01-20 US disclosed
US-5707966-A Antithrombotic agents ELI LILLY AND COMPANY (US) 1998-01-13 US disclosed
US-5705487-A PEPTIDE DERIVATIVES ELI LILLY AND COMPANY (US) 1998-01-06 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed