SCHEMBL7339167

SCHEMBL7339167

CC(C)CC(N)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)N1CCN(c2ccc(F)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
POLB P06746 2/20 0.53
MAPT P10636 1/20 0.49
GPR34 Q9UPC5 2/20 0.48
MME P08473 2/20 0.47
ACE P12821 2/20 0.47
CPA1 P15085 2/20 0.47
ACE2 Q9BYF1 2/20 0.47
CACNA1B Q00975 1/20 0.47
CTSL P07711 1/20 0.46
P2RX7 Q99572 2/20 0.46
YAP1 P46937 1/20 0.45
IL1RN P18510 1/20 0.45
ERAP2 Q6P179 1/20 0.45
ERAP1 Q9NZ08 1/20 0.45
GFER P55789 1/20 0.45
FFAR1 O14842 1/20 0.45
GRM5 P41594 1/20 0.44
MMP1 P03956 1/20 0.44
MMP3 P08254 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337785 0.93 MMP1 (0.52) KDM4EPOLBMAPTMMEACE
SCHEMBL7336001 0.88 CACNA1B (0.52) KDM4EPOLBMAPTMMEACE
SCHEMBL7343237 0.88 CACNA1B (0.60) KDM4EPOLBMAPTCACNA1BCTSL
SCHEMBL7348697 0.87 CACNA1B (0.51) MMEACECPA1ACE2CACNA1B
SCHEMBL7341217 0.87 TACR2 (0.50) MAPTMMEACECPA1ACE2
SCHEMBL7340762 0.86 CACNA1B (0.59) MMEACECPA1ACE2CACNA1B
SCHEMBL7343415 0.86 FAAH (0.52) KDM4EMMEACECPA1ACE2
SCHEMBL7339842 0.86 CACNA1B (0.52) KDM4EPOLBMMEACECPA1
SCHEMBL7338706 0.85 CACNA1B (0.49) MMEACECPA1ACE2CACNA1B
SCHEMBL7337880 0.84 CACNA1B (0.53) MMEACECPA1ACE2CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US claimed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed