SCHEMBL7340283

SCHEMBL7340283

CCOCCOC(=O)C1=C(C)NC(C)=C(C(=O)OCC)C1c1cccc2nsnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 6/20 0.47
KDM4E B2RXH2 6/20 0.47
CYP1A2 P05177 5/20 0.47
CYP3A4 P08684 5/20 0.47
CYP2C19 P33261 5/20 0.47
ALDH1A1 P00352 5/20 0.47
HSD17B10 Q99714 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
GAA P10253 3/20 0.47
LMNA P02545 3/20 0.47
ADORA3 P0DMS8 3/20 0.47
TSHR P16473 3/20 0.47
HIF1A Q16665 2/20 0.47
CYP2D6 P10635 2/20 0.47
NR1I2 O75469 2/20 0.47
ABCB11 O95342 2/20 0.47
NR3C1 P04150 2/20 0.47
TBXA2R P21731 2/20 0.47
OPRK1 P41145 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340826 0.86 CACNA1C (0.51) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL10914306 0.84 CYP2C9 (0.46) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL7342966 0.84 CACNA1C (0.62) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL10914016 0.84 GAA (0.47) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL10913383 0.84 GAA (0.47) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL7340281 0.83 CYP2C9 (0.50) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL10915270 0.82 KDM4E (0.45) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL7348362 0.81 CYP2C9 (0.58) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL7348714 0.80 CYP2C9 (0.69) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19
SCHEMBL11060276 0.78 ALDH1A1 (0.44) CYP2C9KDM4ECYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4466972-A HYPOTENSIVE, ANTIISCHEMIC, ANTISPASMODIC AGENTS SANDOZ LTD. (CH) 1984-08-21 US claimed