SCHEMBL7340301

SCHEMBL7340301

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2C(=O)c3ccccc3C2=O)C1c1ccccn1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.67
KDM4E B2RXH2 4/20 0.67
CASP1 P29466 3/20 0.61
ALDH1A1 P00352 4/20 0.54
CASP7 P55210 1/20 0.51
GAA P10253 4/20 0.50
HPGD P15428 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MAPK1 P28482 1/20 0.47
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GLA P06280 2/20 0.46
BRCA1 P38398 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
CACNA1F O60840 1/20 0.43
CACNA1D Q01668 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7158385 0.83 KDM4E (0.79) HSD17B10KDM4ECASP1ALDH1A1CASP7
SCHEMBL10860930 0.83 KDM4E (0.79) HSD17B10KDM4ECASP1ALDH1A1CASP7
SCHEMBL7350838 0.83 HSD17B10 (0.63) HSD17B10KDM4ECASP1ALDH1A1CASP7
SCHEMBL7343740 0.82 HSD17B10 (0.65) HSD17B10KDM4EALDH1A1GAAHPGD
SCHEMBL7344603 0.82 KDM4E (0.67) HSD17B10KDM4ECASP1ALDH1A1CASP7
SCHEMBL7158896 0.82 KDM4E (0.90) HSD17B10KDM4ECASP1ALDH1A1CASP7
SCHEMBL7160171 0.82 KDM4E (1.00) HSD17B10KDM4ECASP1ALDH1A1CASP7
SCHEMBL7348263 0.81 HSD17B10 (0.66) HSD17B10KDM4EALDH1A1GAAHPGD
SCHEMBL7344861 0.81 HSD17B10 (0.66) HSD17B10KDM4EALDH1A1GAAHPGD
SCHEMBL7343943 0.81 HSD17B10 (0.66) HSD17B10KDM4EALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed