SCHEMBL7340549

SCHEMBL7340549

C#CC[C@H](NC(=O)CNC(=O)c1cccc(NC(=N)N2CCCC2)c1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.41
ITGA5 P08648 1/20 0.41
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TSHR P16473 1/20 0.39
CHRM3 P20309 1/20 0.38
EPHX2 P34913 2/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
HTT P42858 1/20 0.37
GPR139 Q6DWJ6 2/20 0.37
NAMPT P43490 1/20 0.37
PREP P48147 1/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6777651 1.00 ITGB1 (0.41) ITGB1ITGA5KMT2AKDM4ETSHR
SCHEMBL6777468 0.84 ITGB3 (0.44) ITGB1ITGA5KMT2AATML3MBTL1
SCHEMBL6783130 0.82 ITGB1 (0.43) ITGB1ITGA5KMT2AATML3MBTL1
SCHEMBL6773413 0.78 ITGB3 (0.46) ITGB1ITGA5KMT2ATSHRL3MBTL1
SCHEMBL6776549 0.78 ITGB1 (0.42) ITGB1ITGA5KMT2AATML3MBTL1
SCHEMBL6777344 0.77 ITGB1 (0.51) ITGB1ITGA5KMT2AATML3MBTL1
SCHEMBL7340558 0.77 EPHX2 (0.39) KMT2AKDM4ETSHREPHX2ATM
SCHEMBL6774120 0.76 ITGB3 (0.47) ITGB1ITGA5
SCHEMBL8395852 0.75 MAPK1 (0.55) KMT2ACHRM3L3MBTL1HTT
SCHEMBL6776873 0.75 MEN1 (0.44) ITGB1ITGA5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed