SCHEMBL7340552

SCHEMBL7340552

COc1c(C(=O)c2ccccc2OCCCNC(=O)OC(C)(C)C)ccc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCC(O)CC2)c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.36
CDK4 P11802 3/20 0.36
CCND1 P24385 3/20 0.36
CDK2 P24941 3/20 0.36
SIGMAR1 Q99720 2/20 0.35
DRD2 P14416 5/20 0.34
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
SUV39H2 Q9H5I1 1/20 0.33
MAPT P10636 4/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TP53 P04637 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31
HSP90AA1 P07900 1/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339161 0.95 CDK1 (0.35) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7337098 0.94 CDK1 (0.36) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7342217 0.93 SIGMAR1 (0.37) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7343781 0.92 SIGMAR1 (0.35) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7778599 0.91 SIGMAR1 (0.37) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7347827 0.89 MAPT (0.36) DRD2MAPTLMNAHTTSMN1; SMN2
SCHEMBL7340457 0.87 CDK1 (0.35) CDK1CDK4CCND1CDK2DRD2
SCHEMBL7338860 0.87 SIGMAR1 (0.37) SIGMAR1DRD2SUV39H2MAPTTP53
SCHEMBL7345518 0.87 SIGMAR1 (0.38) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7348272 0.86 HDAC3 (0.35) DRD2MAPTLMNAHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed