SCHEMBL7339161

SCHEMBL7339161

COc1c(C(=O)c2ccccc2OCCCNC(=O)OC(C)(C)C)ccc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCC(N(C)C)CC2)c1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.35
CDK4 P11802 3/20 0.35
CCND1 P24385 3/20 0.35
CDK2 P24941 3/20 0.35
SIGMAR1 Q99720 2/20 0.34
DRD2 P14416 4/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
SMO Q99835 1/20 0.33
SUV39H2 Q9H5I1 1/20 0.33
ABL1 P00519 1/20 0.31
FYN P06241 1/20 0.31
SRC P12931 1/20 0.31
PTK6 Q13882 1/20 0.31
MAPT P10636 3/20 0.31
LMNA P02545 2/20 0.31
HTT P42858 2/20 0.31
AVPR2 P30518 1/20 0.31
AVPR1A P37288 1/20 0.31
AVPR1B P47901 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7337098 0.95 CDK1 (0.36) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7340552 0.95 CDK1 (0.36) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7340457 0.93 CDK1 (0.35) CDK1CDK4CCND1CDK2DRD2
SCHEMBL7342217 0.92 SIGMAR1 (0.37) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7343781 0.92 SIGMAR1 (0.35) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL8673452 0.91 MEN1 (0.34) SIGMAR1DRD2SUV39H2
SCHEMBL7778599 0.90 SIGMAR1 (0.37) CDK1CDK4CCND1CDK2SIGMAR1
SCHEMBL7347827 0.88 MAPT (0.36) DRD2MAPTLMNAHTTSMN1; SMN2
SCHEMBL7338860 0.87 SIGMAR1 (0.37) SIGMAR1DRD2SUV39H2MAPTAVPR2
SCHEMBL7345518 0.86 SIGMAR1 (0.38) CDK1CDK4CCND1CDK2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-B1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2001-09-05 EP disclosed
WO-1996041795-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-12-27 WO disclosed