SCHEMBL7340574

SCHEMBL7340574

Cc1cc2c(c(C(=O)C(C)CC(=O)O)c1)OCCN2

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HSD17B10 Q99714 1/20 0.37
RET P07949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7349907 0.88 ALDH1A1 (0.35) ALDH1A1GAAMAPTHSD17B10RET
SCHEMBL7345073 0.86 ALDH1A1 (0.34) ALDH1A1GAAMAPTHSD17B10RET
SCHEMBL7342732 0.80 MMP2 (0.40)
SCHEMBL7344276 0.80 PDE3B (0.42)
SCHEMBL7338777 0.72 ALDH1A1 (0.47) ALDH1A1GAAMAPTHSD17B10
SCHEMBL12116975 0.68 ALDH1A1 (0.50) ALDH1A1GAAMAPTHSD17B10RET
SCHEMBL4967534 0.67 ALDH1A1 (0.53) ALDH1A1GAAMAPTHSD17B10RET
SCHEMBL4481502 0.65 ALDH1A1 (0.50) ALDH1A1GAAMAPTHSD17B10RET
SCHEMBL21316386 0.64 ADORA2A (0.38) ALDH1A1GAAMAPTHSD17B10
SCHEMBL7275955 0.64 AKR1C4 (0.39) ALDH1A1MAPTHSD17B10RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509845-A1 (+) and (-) enantiomers of 5-aliphatic-6-(benzoxazinyl- or benzothiazinyl)-2,3,4,5-tetrahydropyridazin-3-ones ORTHO PHARMACEUTICAL CORPORATION (US) 1992-10-21 EP disclosed
US-5081242-A Cardiotonic and bronchodilator agents; phosphodiesterase inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1992-01-14 US disclosed
US-4766118-A CARDIOTONIC AGENTS, PHOSPHODIESTERASE INHIBITORS ORTHO PHARMACEUTICAL CORPORATION (US) 1988-08-23 US disclosed
EP-0272914-A2 6-Benzoxazinyl- and 6-benzothiazinyl-2,3,4,5-tetrahydropyridazin-3-ones ORTHO PHARMACEUTICAL CORPORATION (US) 1988-06-29 EP disclosed
US-4721784-A MUSCLE RELAXANTS, BRONCHODILATOR AGENTS, CARDIOTONIC AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1988-01-26 US disclosed