SCHEMBL7340645

SCHEMBL7340645

O=C(O)CCC1(NC(=O)CNC(=O)c2cccc(NC(=O)NCc3ccccc3)c2)C=CC=NC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
KDR P35968 1/20 0.41
MAPK1 P28482 2/20 0.40
LMNA P02545 1/20 0.40
SENP1 Q9P0U3 2/20 0.39
PPARG P37231 1/20 0.39
TSHR P16473 1/20 0.39
MAPK14 Q16539 1/20 0.39
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
KMT2A Q03164 1/20 0.38
ROCK2 O75116 1/20 0.38
GRK2 P25098 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NAMPT P43490 3/20 0.37
EGLN2 Q96KS0 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7374315 0.94 NAMPT (0.45) HTTTSHRKMT2AROCK2GRK2
SCHEMBL7347133 0.93 ALDH1A1 (0.41) ALDH1A1HPGDHTTMAPK1LMNA
SCHEMBL7349095 0.83 KMT2A (0.40) ALDH1A1MAPK14RAB9ANPC1MITF
SCHEMBL7338423 0.82 NAMPT (0.41) ALDH1A1HPGDHTTLMNATSHR
SCHEMBL7338453 0.79 KMT2A (0.42) HPGDLMNAMITFKMT2A
SCHEMBL7341050 0.77 ALDH1A1 (0.37) ALDH1A1LMNATSHRRAB9ANPC1
SCHEMBL6776908 0.77 MAPK1 (0.50) ALDH1A1HPGDHTTKDRMAPK1
SCHEMBL7348795 0.74 PPARG (0.43) ALDH1A1HPGDHTTKDRMAPK1
Chlorobenzene SCHEMBL7832714 0.73 KDM4E (0.52) ALDH1A1HTTKDRMAPK1LMNA
SCHEMBL6773426 0.72 MAPK1 (0.45) ALDH1A1HPGDHTTKDRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed