SCHEMBL7340836

SCHEMBL7340836

CCOC(=O)CCCNc1c(C)cccc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.58
USP2 O75604 1/20 0.53
HSD17B10 Q99714 1/20 0.53
NLRP3 Q96P20 3/20 0.47
PDE5A O76074 1/20 0.46
ELANE P08246 1/20 0.46
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
POLB P06746 1/20 0.43
KDM4E B2RXH2 3/20 0.43
LTA4H P09960 1/20 0.43
MAPT P10636 1/20 0.43
NPC1 O15118 1/20 0.41
MEN1 O00255 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11311241 0.89 TOP2A (0.63) TOP2AUSP2HSD17B10NLRP3PDE5A
SCHEMBL11325006 0.84 NLRP3 (0.58) TOP2AUSP2HSD17B10NLRP3PDE5A
SCHEMBL28859305 0.83 POLB (0.50) HSD17B10ALDH1A1CYP3A4POLBKDM4E
SCHEMBL28278344 0.82 CA12 (0.49) HSD17B10ALDH1A1POLBKDM4E
SCHEMBL5136112 0.81 CA12 (0.48) HSD17B10ALDH1A1POLBKDM4E
SCHEMBL9830020 0.80 TOP2A (0.61) TOP2AUSP2HSD17B10NLRP3ALDH1A1
SCHEMBL11312355 0.79 TOP2A (0.61) TOP2AUSP2HSD17B10NLRP3PDE5A
SCHEMBL3668324 0.78 TOP2A (0.60) TOP2AUSP2HSD17B10PDE5AELANE
SCHEMBL25142537 0.77 ALDH1A1 (0.49) TOP2AUSP2HSD17B10PDE5AELANE
SCHEMBL13073786 0.77 POLB (0.56) HSD17B10ALDH1A1CYP3A4POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022282-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1996-07-25 WO disclosed