SCHEMBL7340883

SCHEMBL7340883

N=C(N)N1CCC(CN[C@H](Cc2ccccc2)C(=O)N2CCC[C@H]2C(N)=O)CC1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 0.56
F2 P00734 4/20 0.56
ACE P12821 1/20 0.52
OPRM1 P35372 1/20 0.46
TRHR P34981 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299051 1.00 PRSS1 (0.56) PRSS1F2ACEOPRM1TRHR
SCHEMBL7299046 1.00 PRSS1 (0.56) PRSS1F2ACEOPRM1TRHR
SCHEMBL7295808 0.91 F2 (0.52) PRSS1F2ACEOPRM1
SCHEMBL7050971 0.91 F2 (0.52) PRSS1F2ACEOPRM1
SCHEMBL7113615 0.91 F2 (0.52) PRSS1F2ACEOPRM1
SCHEMBL7303710 0.86 YAP1 (0.51) PRSS1F2ACE
SCHEMBL8072498 0.84 ACE (0.57) ACEOPRM1
SCHEMBL7346744 0.81 F2 (0.54) PRSS1F2
SCHEMBL7338542 0.81 F2 (0.54) PRSS1F2
SCHEMBL7340878 0.80 F2 (0.60) PRSS1F2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0601459-A2 Sulfonamido heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-06-15 EP disclosed