SCHEMBL8072498

SCHEMBL8072498

CCN[C@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ACE P12821 7/20 0.57
ACE2 Q9BYF1 4/20 0.51
OPRM1 P35372 1/20 0.51
LTA4H P09960 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299046 0.84 PRSS1 (0.56) ACEOPRM1
SCHEMBL7340883 0.84 PRSS1 (0.56) ACEOPRM1
SCHEMBL7299051 0.84 PRSS1 (0.56) ACEOPRM1
SCHEMBL5710967 0.83 ACE (0.61) ACEACE2OPRM1LTA4H
SCHEMBL7280460 0.83 ACE (0.69) ACEACE2OPRM1
SCHEMBL7343554 0.82 ACE (0.51) ACEACE2OPRM1LTA4H
SCHEMBL8250626 0.82 OPRM1 (0.60) ACEOPRM1
SCHEMBL6412059 0.81 ACE (0.66) ACE
SCHEMBL7087290 0.81 ACE (0.66) ACE
SCHEMBL6412055 0.81 ACE (0.66) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1012165-A1 PROCESS FOR THE PREPARATION OF N-METHYL-D-PHENYLALANYL-N- 1- 3- (AMINOIMINOMETHYL)AMINO]PROPYL]-3,3-DIFLUORO-2-OXOHEXYL]-L-PROLINAMIDE Aventis Pharmaceuticals Inc. (US) 2000-06-28 EP claimed
WO-1997035874-A1 PROCESS FOR THE PREPARATION OF N-METHYL-D-PHENYLALANYL-N-[1-[3-[(AMINOIMINOMETHYL)AMINO]PROPYL]-3,3-DIFLUORO-2-OXOHEXYL]-L-PROLINAMIDE HOECHST MARION ROUSSEL, INC. (US) 1997-10-02 WO claimed