SCHEMBL7340989

SCHEMBL7340989

C=CC([C]=O)c1ccc(OCC)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 9/20 0.47
NQO1 P15559 1/20 0.47
LTA4H P09960 1/20 0.41
TSHR P16473 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HPGD P15428 1/20 0.40
LMNA P02545 1/20 0.40
PARP10 Q53GL7 1/20 0.39
RELA Q04206 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CNR2 P34972 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6708195 0.77 NQO1 (0.56) ACACBNQO1LTA4HTSHRTDP1
SCHEMBL910341 0.75 NQO1 (0.54) ACACBNQO1TSHRTDP1HPGD
SCHEMBL8068074 0.74 NQO1 (0.52) ACACBNQO1LTA4HTSHRTDP1
SCHEMBL13278546 0.73 NQO1 (0.47) ACACBNQO1LTA4HTSHRTDP1
SCHEMBL7438043 0.71 ACACB (0.42) ACACBNQO1TSHRTDP1CNR2
SCHEMBL367639 0.70 CYP2C19 (0.38) TSHRTDP1HPGDLMNAMAPT
SCHEMBL2490798 0.69 NQO1 (0.70) ACACBNQO1LTA4HTSHRTDP1
SCHEMBL824979 0.69 NQO1 (0.70) ACACBNQO1LTA4HTSHRTDP1
1,4-Diethoxybenzene SCHEMBL9651064 0.69 NQO1 (0.70) NQO1LTA4HTSHRTDP1LMNA
SCHEMBL15330491 0.69 NQO1 (0.56) ACACBNQO1LTA4HTSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5459142-A Autoimmune disease, atherosclerosis, antiischemic agents and nephritis OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-17 US disclosed
EP-0511879-B1 Pyrazine derivatives OTSUKA PHARMA CO LTD (JP) 1995-03-22 EP disclosed
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed
US-4514401-A CARDIOTONICS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1985-04-30 US disclosed
US-4487772-A CARDIOTONIC AGENTS OTSUKA PHARMACEUTICAL CO. LTD. (JP) 1984-12-11 US disclosed
US-4468402-A Carbostyril derivatives, process for producing the same and cardiotonic compositions containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-08-28 US disclosed
US-4454130-A CARDIOTONIC, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1984-06-12 US disclosed