SCHEMBL7341880

SCHEMBL7341880

CCc1[nH]c(=O)[nH]c1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.53
PDE3A Q14432 2/20 0.53
JAK2 O60674 1/20 0.45
THRB P10828 1/20 0.45
LMNA P02545 1/20 0.43
PDE4A P27815 12/20 0.42
PDE4B Q07343 12/20 0.42
PDE4C Q08493 12/20 0.42
PDE4D Q08499 12/20 0.42
HCAR2 Q8TDS4 2/20 0.41
DHODH Q02127 1/20 0.40
NSD2 O96028 1/20 0.38
ABL1 P00519 1/20 0.38
GAA P10253 1/20 0.38
IDE P14735 1/20 0.38
RIN1 Q13671 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10811057 0.81 PDE3B (0.51) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL11186838 0.80 JAK2 (0.47) PDE3BPDE3AJAK2THRBLMNA
SCHEMBL10632760 0.79 PDE3B (0.70) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10968412 0.78 JAK2 (0.45) PDE3BPDE3AJAK2THRBLMNA
SCHEMBL10811069 0.78 PDE3B (0.49) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL9786614 0.78 PDE3B (0.49) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10805601 0.76 PDE3B (0.47) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL256096 0.76 MAPT (0.56) PDE3BPDE3ALMNAABL1GAA
SCHEMBL22783664 0.75 JAK2 (0.61) JAK2THRBLMNADHODHNSD2
SCHEMBL22766845 0.75 PDE3B (0.46) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169164-B1 IMIDAZOLONECARBONYLARYLIMIDAZOLES; METHOD OF MANUFACTURE, METHOD OF USE AND COMPOSITIONS USEFUL THEREOF SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-31 EP disclosed
US-4709043-A Process for the preparation of imidazolonecarbonylarylimidazoles SCHERING A.G. (DE) 1987-11-24 US disclosed
EP-0169164-A1 Imidazolonecarbonylarylimidazoles; method of manufacture, method of use and compositions useful thereof SCHERING AKTIENGESELLSCHAFT (DE) 1986-01-22 EP disclosed
US-4556665-A Cardiotonic 1,3-dihydro-4-[[(imidazol-1-yl)aryl]carbonyl]imidazol-2-ones SCHERING A.G. (DE) 1985-12-03 US disclosed