SCHEMBL7345217

SCHEMBL7345217

Cc1ccc(NCC(=O)Oc2ccccc2)c(CCC(=O)OC(C)(C)C)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
CREBBP Q92793 1/20 0.35
KMT2A Q03164 3/20 0.34
KDM4E B2RXH2 3/20 0.34
GAA P10253 2/20 0.34
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
GLA P06280 1/20 0.34
HIF1A Q16665 1/20 0.34
LIPG Q9Y5X9 1/20 0.33
MEN1 O00255 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
BRD4 O60885 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
AKT1 P31749 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7347509 0.71 MAPKAPK2 (0.37) KDM4EALDH1A1HPGDGLAMAPKAPK2
SCHEMBL5849169 0.71 EPHX2 (0.50) TSHRKMT2AKDM4EGAAMAPT
SCHEMBL7117442 0.69 ELANE (0.44) KMT2AKDM4EMAPTALDH1A1RAB9A
SCHEMBL6779226 0.68 KMT2A (0.34) KMT2AKDM4EMAPTALDH1A1MEN1
SCHEMBL7434663 0.67 ALDH1A1 (0.42) KMT2AKDM4EGAAMAPTALDH1A1
SCHEMBL6178813 0.66 RAB9A (0.50) TSHRKMT2AGAAMAPTMEN1
SCHEMBL6775183 0.66 KMT2A (0.44) KMT2AKDM4EALDH1A1GLAMEN1
SCHEMBL27561944 0.66 EPHX2 (0.46) KMT2AKDM4EGAAMAPTALDH1A1
SCHEMBL6437790 0.66 MAPT (0.47) KDM4EGAAMAPTALDH1A1HPGD
SCHEMBL2001318 0.65 GAA (0.59) TSHRKMT2AKDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed