SCHEMBL7345498

SCHEMBL7345498

CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cccc(Br)c1.c1ccc2c(c1)CNC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.64
POLB P06746 2/20 0.61
HIF1A Q16665 5/20 0.58
CYP2C9 P11712 5/20 0.58
MEN1 O00255 4/20 0.58
CYP1A2 P05177 4/20 0.58
CYP3A4 P08684 4/20 0.58
CYP2C19 P33261 4/20 0.58
KMT2A Q03164 4/20 0.58
MAPT P10636 3/20 0.58
TSHR P16473 3/20 0.58
LMNA P02545 2/20 0.58
CYP2D6 P10635 2/20 0.58
NFKB1 P19838 2/20 0.58
THPO P40225 2/20 0.58
MAPK1 P28482 1/20 0.58
GPR55 Q9Y2T6 1/20 0.58
CACNA1B Q00975 1/20 0.55
CACNA1F O60840 4/20 0.52
CACNA1D Q01668 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343711 0.88 ADORA3 (0.64) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL7341782 0.88 CACNA1D (0.67) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL7349302 0.88 ADORA3 (0.64) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL3032551 0.86 CACNA1F (0.66) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL7349506 0.85 CACNA1F (0.68) ADORA3POLBHIF1ACYP2C9MEN1
Nitrendipine SCHEMBL7343607 0.85 HIF1A (0.83) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL29676320 0.84 TSHR (0.69) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL3326231 0.84 TSHR (0.69) ADORA3POLBHIF1ACYP2C9MEN1
SCHEMBL7343550 0.82 ADORA3 (0.58) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7347764 0.82 ADORA3 (0.64) ADORA3POLBHIF1ACYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed